
个人简历
车志平,男,生于1984年11月,甘肃天水人,中共党员,博士,教授,博导。
E-mail:zhipingche@163.com
联系电话:15037996651
办公地点:园艺与植物保护学院114室
研究领域:
1. 植物源农用活性化合物结构优化、构效关系及作用机理研究
2. 基于植物源农用活性化合物为先导的新农药半合成研究
研究生招生:
1. 学术学位:植物保护
2. 专业学位:资源利用与植物保护
一、教学及科研情况简介
主持国家自然科学基金、河南省科技攻关、河南省高等学校青年骨干教师、河洛青年人才托举工程、校青年学术带头人等科研项目10余项。现为《Advanced Science》、《Journal of Agricultural and Food Chemistry》和《Industrial Crops and Products》等多个TOP期刊的审稿专家;以第一或通讯作者在《Journal of Agricultural and Food Chemistry》、《Pest Management Science》和《Industrial Crops and Products》等TOP期刊发表学术论文60余篇;授权发明专利20余件,成果转化30余万元;获省部级奖励3项。入选河南省高等学校青年骨干教师、河洛青年人才、校青年学术带头人;当选河南省科协评审咨询专家,河南省高新技术企业评审专家,洛阳市科普专家,洛阳市科协工作先进个人;获河南省优秀学士学位论文指导教师,校教学标兵、优秀教师、优秀党员、优秀学业导师、优秀辅导教师等荣誉称号。讲授“植物化学保护学”、“农药加工与管理”、“农药生物测定”等本科生课程,“农药药理学”、“农药化学”、“绿色农药研究及应用技术”等研究生课程。
二、教育背景及工作经历
1. 2024.01-至今,河南科技大学,园艺与植物保护学院,教授,科研秘书
2. 2020.09-2023.12,河南科技大学,园艺与植物保护学院,副教授,科研秘书
3. 2018.01-2020.09,河南科技大学,林学院植物保护系,副教授
4. 2013.07-2017.12,河南科技大学,园艺与植物保护学院,讲师
5. 2010.09-2013.06,西北农林科技大学,化学生物学专业,理学博士
6. 2007.09-2010.06,西北农林科技大学,农药学专业,农学硕士
7. 2003.09-2007.06,河南科技大学,植物保护专业,农学学士
三、个人荣誉
2017年获河南科技大学“优秀教师”称号;
2018年获河南科技大学“SRTP”优秀指导教师称号;
2018年获“河南省优秀科技特派员”称号;
2019年获河南科技大学“SRTP”优秀指导教师称号;
2019年获第十四届“挑战杯”河南省二等奖指导老师称号;
2019年获河南科技大学理论教学“二等奖”称号;
2019年获河南科技大学“优秀共产党员”称号;
2020年获河南科技大学“优秀学业导师”称号;
2021年获河南科技大学“优秀学业导师”称号;
2021年入选河南省科研设施与仪器共享服务平台“高级培训师”;
2022年获河南科技大学“SRTP”优秀指导教师称号;
2022年入选“河南省科协评审咨询专家”;
2023年获河南科技大学“优秀辅导教师”称号;
2023年入选“河南省高新技术企业专家库评审专家”;
2023年获河南科技大学2023届本科毕业论文“一等奖优秀指导教师”称号;
2023年获河南科技大学“教学标兵”称号;
2023年入选洛阳市科学技术协会“科技创新智库专家”;
2023年获“河洛青年人才”称号;
2023年获栾川县“科技创新工作先进个人”称号;
2023年获洛阳市“科协工作先进个人”称号;
2023年入选首批“洛阳市科普专家”;
2023年获第十六届“挑战杯”河南省二等奖指导教师称号;
2024年获河南科技大学“SRTP”优秀指导教师称号;
2024年获“河南省高等学校青年骨干教师”称号;
2024年获“河南省优秀学士学位论文”指导教师称号。
四、科研项目
1. 国家自然科学基金联合项目(U1604105),2017.01-2019.12,结题,主持;
2. 河南省科技攻关项目(202102110068),2020.01-2021.12,结题,主持;
3. 河南省高等学校青年骨干教师培养计划项目(2020GGJS080),2021.01-2023.12,结题,主持;
4. 河洛青年人才托举工程项目(2023HLTJ01),2023.09-2024.12,结题,主持;
5. 河南省科技特派员项目(2018SQ090),2018.07-2024.04,结题,主持;
6. 河南科技大学青年学术带头人项目(13490003),2017.03-2020.03,结题,主持;
7. 河南科技大学高级别培育基金项目(2015GJB024),2015.01-2016.12,结题,主持;
8. 河南科技大学博士科研启动项目(09001763),2014.01-2016.12,结题,主持。
9. 河南省自然科学基金面上项目(182300410016),2018.01-2019.12,结题,第一参与人;
10. 河南省科技攻关项目(182102110202),2018.01-2019.12,结题,第一参与人;
11. 河南省科技攻关项目(222102110023),2022.01-2023.12,结题,第一参与人;
12. 河南省科技攻关项目(252102111103),2025.01-2026.12,在研,第一参与人。
五、学术论文
1. Liu Yibo, Tian Yuee, Peng Hong, Zhang Fulong, Huang Xiaobo, Chen Genqiang, Zhou Lin, Che Zhiping(通讯作者), Design, synthesis, and anti-oomycete and antifungal activities of novel paeonol derivatives containing a pyrazole ring, Journal of Agricultural and Food Chemistry, 2025, 73(16): 9533-9540.(中科院一区,Top期刊)
2. Huang Xiaobo, Hao Nan, Shu Lili, Wei Zhenyang, Shi Jiawei, Tian Yuee, Chen Genqiang, Yang Xinling, Che Zhiping(通讯作者), Preparation and insecticidal activities of betulin-cinnamic acid-related hybrid compounds and insights into the stress response of Plutella xylostella L., Pest Management Science, 2025, DOI: 10.1002/ps.8785.(中科院一区,Top期刊)
3. Hu Mei, Guo Xiaolong, Tian Yuee, Li Yan, Liu Yibo, Huang Xiaobo, Chen Genqiang, Che Zhiping(通讯作者), Synthesis of paeonol hydrazone derivatives and their anti-oomycete, anti-fungal, and nematicidal activities, Pest Management Science, 2024, 80(11): 5746-5758.(中科院一区,Top期刊)
4. Tian Yuee, Yin Wanying, Wang Ruiguang, Sun Huilu, Xu Shaobin, Huang Xiaobo, Chen Genqiang, Che Zhiping(通讯作者), Non-food renewable and bioactive products for pesticides: synthesis, anti-oomycete and anti-fungal activities of 9R-acyloxyquinine derivatives bearing an 1,3,4-oxadiazole moiety, Industrial Crops & Products, 2024, 222, 119751.(中科院一区,Top期刊)
5. Che Zhiping(第一且通讯作者), Guo Xiaolong, Li Yuanhao, Zhang Song, Zhu Lina, He Jiaxuan, Sun Di, Guo Yihao, Liu Yibo, Wei Ruxue, Huang Xiaobo, Liu Shengming, Chen Genqiang, Tian Yuee, Synthesis of paeonol ester derivatives and their insecticidal, nematicidal, and anti-oomycete activities, Pest Management Science, 2022, 78(8): 3442-3455.(中科院一区,Top期刊)
6. Huang Xiaobo, Hao Nan, Wang Qun, Li Ruru, Zhang Ge, Chen Genqiang, Liu Shengming, Che Zhiping(通讯作者), Non-food bioactive forest product liriodenine: sources, chemistry, and bioactivities, Industrial Crops and Products, 2022, 187: 115447.(中科院一区,Top期刊)
7. Huang Xiaobo, Hao Nan, Chen Genqiang, Liu Shengming, Che Zhiping(通讯作者), Chemistry and biology of nuciferine, Industrial Crops and Products, 2022, 179: 114694.(中科院一区,Top期刊)
8. Che Zhiping(第一作者), Yu Xiang, Zhi Xiaoyan, Fan Lingling, Yao Xiaojun, Xu Hui, Synthesis of novel 4α-(acyloxy)-2'(2',6')-(di)halogenopodophyllotoxin derivatives as insecticidal agents, Journal of Agricultural and Food Chemistry, 2013, 61(34): 8148-8155.(中科院一区,Top期刊)
9. Che Zhiping(第一作者), Zhang Shaoyong, Shao Yonghua, Fan Lingling, Xu Hui, Yu Xiang, Zhi Xiaoyan, Yao Xiaojun, Zhang Rui, Synthesis and quantitative structure-activity relationship (QSAR) study of novel N-arylsulfonyl-3-acylindole arylcarbonyl hydrazone derivatives as nematicidal agents, Journal of Agricultural and Food Chemistry, 2013, 61(24): 5696-5705.(中科院一区,Top期刊)
10. Yang Ruige, Huang Xiaobo, Che Zhiping(共同第一作者), Zhang Yuanyuan, Xu Hui, Application of sustainable natural resources in crop protection: Podophyllotoxin-based botanical pesticides derived from Podophyllum hexandrum for controlling crop-threatening insect pests, Industrial Crops & Products, 2017, 107: 45-53.(中科院一区,Top期刊)
11. Yin Wanying, Tian Yuee, Ma Shiyue, Guo Xiaolong, Wang Ruiguang, Liu Yibo, Huang Xiaobo, Chen Genqiang, Che Zhiping(通讯作者), Synthesis, anti-oomycete and anti-fungal activities of aminoguanidine derivatives of paeonol sulfonate, Journal of Molecular Structure, 2025, 1321, 140085.(中科院二区)
12. Che Zhiping(第一且通讯作者), Zhang Song, Guo Yihao, Liu Yibo, Wei Ruxue, Zhou Lin, Huang Xiaobo, Liu Shengming, Chen Genqiang, Tian Yuee, Synthesis, anti-oomycete and anti-fungal activities of novel cinchona alkaloid derivatives bearing carbamate moiety, Journal of Molecular Structure, 2023, 1291, 136055.(中科院二区)
13. Che Zhiping(第一且通讯作者), Guo Xiaolong, Huang Xiaobo, Wang Tiewei, Zhou Lin, Liu Shengming, Chen Genqiang, Tian Yuee, Synthesis, anti-oomycete activity of 1-sulfonyloxy/acyloxysesamol derivatives, Journal of Molecular Structure, 2023, 1283, 135260.(中科院二区)
14. Tian Yuee, Li Yan, Wang Shuhe, He Jiaxuan, Sun Di, Liu Shengming, Chen Genqiang, Che Zhiping(通讯作者), Genome sequence resource and annotation of Calonectria montana, an economically important pathogen with a broad host range, Molecular Plant-Microbe Interactions, 2022, 35(6): 492-495.(中科院二区)
15. Tian Yuee, Li Yan, Wang Shuhe, Ren Yingge, He Yilin, Chen Genqiang, Che Zhiping(通讯作者), Whole-genome sequence resource and annotation of Cladosporium paeoniae, the causal pathogen of tree peony leaf mold, Molecular Plant-Microbe Interactions, 2022, 35(11): 1048-1051.(中科院二区)
16. Che Zhiping(第一且通讯作者), Tian Yuee, Liu Shengming, Jiang Jia, Hu Mei, Chen Genqiang, Microwave-assisted expeditious synthesis of 2-alkyl-2-(N-arylsulfonylindol-3-yl)-3-N-acyl-5-aryl-1,3,4-oxadiazolines catalyzed by HgCl2 under solvent-free conditions as potential anti-HIV-1 agents, Molecules, 2018, 23(11), 2936.(中科院二区)
17. Yu Xiang, Che Zhiping(共同第一作者), Xu Hui, Recent advances in the chemistry and biology of podophyllotoxins, Chemistry-A European Journal, 2017, 23(19): 4467-4526.(中科院二区)
18. Wang Ruiguang, Li Yuanhao, Yin Wanying, Sun Huilu, Xu Shaobin, Shuang Shaoyan, Tian Yuee, Huang Xiaobo, Chen Genqiang, Che Zhiping(通讯作者), Synthesis, anti-oomycete and anti-fungal activities of anhydride derivatives of oleanolic acid, Chemistry & Biodiversity, 2024, 21(12): e202401952.
19. Huang Xiaobo, Shu Lili, Hao Nan, Wei Zhenyang, Qian Le, Tian Yuee, Cheng Zejun, Chen Genqiang, Liu Shengming, Deng Shuzhen, Guo Yashuang, Che Zhiping(通讯作者), Synthesis and antifungal evaluation of cinnamic acid-geraniol hybrids as potential fungicides, Chemistry & Biodiversity, 2024, 21(12): e202401348.
20. Tian Yuee, Ma Shiyue, Liu Yibo, Li Yan, Chen Genqiang, Che Zhiping(通讯作者), Synthesis of novel 4-acyloxy-2′-bromo-6′-chloropodophyllotoxin derivatives displaying significant insecticidal activity against Mythimna Separata, Chemistry & Biodiversity, 2024, 21(7): e202400929.
21. Zhang Xiaofang, Guo Xiaolong, Yin Wanying, Wang Ruiguang, Tian Yuee, Sun Huilu, Xu Shaobin, Shuang Shaoyan, Huang Xiaobo, Chen Genqiang, Che Zhiping(通讯作者), Synthesis, anti-oomycete and anti-fungal activities of novel paeonol ester derivatives containing a schiff base, Natural Product Research, 2024, DOI: 10.1080/14786419.2024.2426205.
22. Hai Fei, Wei Ruxue, Li Yan, Wang Ruiguang, Tian Yuee, Liu Shengming, Chen Genqiang, Che Zhiping(通讯作者), Combinatorial synthesis of indole derivatives as anti-oomycetes agents, Combinatorial Chemistry & High Throughput Screening, 2024, 27(19): 2816-2823.
23. Guo Yihao, Liu Yibo, Ma Yingying, Li Yan, Tian Yuee, Huang Xiaobo, Qian Le, Liu Shengming, Chen Genqiang, Che Zhiping(通讯作者), Design, synthesis, and anti-oomycete activity of 3-acyloxymaltol/ethyl maltol derivatives, Journal of Asian Natural Products Research, 2024, 26(10): 1166-1174.
24. Wei Ruxue, Liu Yibo, Yin Wanying, Wang Ruiguang, Tian Yuee, Huang Xiaobo, Qian Le, Liu Shengming, Chen Genqiang, Che Zhiping(通讯作者), Design, synthesis and anti-oomycete activity of 2-acyloxyhinokitiol derivatives, Natural Product Research, 2024, DOI: 10.1080/14786419.2024.2331021.
25. Liu Yibo, Li Yan, Tian Yuee, Guo Yihao, Wei Ruxue, Huang Xiaobo, Qian Le, Liu Shengming, Chen Genqiang, Che Zhiping(通讯作者), Synthesis of novel 18β-glycyrrhetinic acid sulfonate derivatives displaying significant anti-oomycete activity against Phytophthora capsici, Natural Product Research, 2023, DOI: 10.1080/14786419.2023.2280999.
26. Zhu Lina, Tian Yuee, Wang Tiewei, Huang Xiaobo, Zhou Lin, Liu Shengming, Chen Genqiang, Che Zhiping(通讯作者), Semisynthesis, anti-oomycete and anti-fungal activities of ursolic acid ester derivatives, Natural Product Research, 2024, 38(6), 906-915.
27. Chen Yingwu, Zhang Song, Tian Yuee, Huang Xiaobo, Zhou Lin, Liu Shengming, Chen Genqiang, Che Zhiping(通讯作者), Synthesis, anti-oomycete and anti-fungal activities of novel cinchona alkaloid derivatives containing sulfonate moiety, Chemistry & Biodiversity, 2023, 20, e202300607.
28. He Jiaxuan, Tian Yuee, Huang Xiaobo, Wang Tiewei, Zhou Lin, Liu Shengming, Chen Genqiang, Che Zhiping(通讯作者), Synthesis, anti-oomycete and fungal activities of resveratrol sulfonate derivatives containing three esters moieties, Journal of Natural Pesticide Research, 2023, 3, 100023.
29. Che Zhiping(第一且通讯作者), Zhang Song, He Jiaxuan, Sun Di, Guo Xiaolong, Li Yuanhao, Zhu Lina, Guo Yihao, Liu Yibo, Tian Yuee, Huang Xiaobo, Liu Shengming, Chen Genqiang, Combinatorial synthesis of sulfonate derivatives of α/β-naphthol as anti-oomycete agents, Combinatorial Chemistry & High Throughput Screening, 2022, 25(12), 2026-2032.
30. Che Zhiping(第一且通讯作者), Liu Yibo, Chen Luyao, Xing Puhou, Li Xiangdong, Huang Xiaobo, Liu Shengming, Chen Genqiang, Lin Xiaomin, Tian Yuee, Synthesis of hinokitiol sulfonate derivatives and their anti-oomycete and nematicidal activities, Chemistry & Biodiversity, 2022, 19(8): e202200580.
31. Xing Puhou, Che Zhiping(通讯作者), Liu Yibo, He Jiaxuan, Wei Ruxue, Chen Luyao, Zhang Song, Huang Xiaobo, Yang Yingjun, Liu Shengming, Chen Genqiang, Tian Yuee, Synthesis and anti-oomycete preliminary mechanism of sulfonate derivatives of ethyl maltol, Chemistry & Biodiversity, 2022, 19(6): e202200255.
32. Che Zhiping(第一且通讯作者), Li Yuanhao, Guo Xiaolong, He Jiaxuan, Zhang Song, Zhu Lina, Liu Yibo, Wei Ruxue, Yang Yingjun, Huang Xiaobo, Liu Shengming, Chen Genqiang, Tian Yuee, Synthesis and anti-oomycete activity of sulfonate derivatives of Fenjuntong, Chemistry & Biodiversity, 2022, 19(4): e202101039.
33. Chen Genqiang, Zhu Lina, Yang Jinming, Zhang Song, Li Yuanhao, Guo Xiaolong, Sun Di, He Jiaxuan, Tian Yuee, Liu Shengming, Jiang Jia, Huang Xiaobo, Che Zhiping(通讯作者), Synthesis of novel 3/5(3,5)-(di)nitropaeonolhydrazone derivatives as nematicidal agents, Journal of Asian Natural Products Research, 2022, 24(1): 66-75.
34. Chen Genqiang, Zhu Lina, He Jiaxuan, Zhang Song, Li Yuanhao, Guo Xiaolong, Sun Di, Tian Yuee, Liu Shengming, Huang Xiaobo, Che Zhiping(通讯作者), Combinatorial synthesis of novel 1-sulfonyloxy/acyloxyeugenol derivatives as fungicidal agents, Combinatorial Chemistry & High Throughput Screening, 2022, 25(9): 1545-1551.
35. Chen Genqiang, Zhu Lina, Xia Yanfei, Yang Jinming, Zhang Song, Li Yuanhao, Guo Xiaolong, Sun Di, He Jiaxuan, Tian Yuee, Liu Shengming, Jiang Jia, Che Zhiping(通讯作者), Combinatorial synthesis of novel 3/5(3,5)-(di)nitro/chloropaeonol carbonyl hydrazone derivatives as nematicidal agents, Combinatorial Chemistry & High Throughput Screening, 2022, 25(6): 1031-1039.
36. Chen Genqiang, Zhu Lina, He Jiaxuan, Zhang Song, Li Yuanhao, Guo Xiaolong, Sun Di, Tian Yuee, Liu Shengming, Huang Xiaobo, Che Zhiping(通讯作者), Synthesis and anti-oomycete activity of 1-sulfonyloxy/acyloxydihydroeugenol derivatives, Chemistry & Biodiversity, 2021, 18(9): e2100329.
37. Chen Genqiang, Sun Di, Yang Jinming, Zhang Song, Tian Yuee, Che Zhiping(通讯作者), Liu Shengming, Jiang Jia, Lin Xiaomin, Synthesis of sulfonate derivatives of carvacrol and thymol as anti-oomycetes agents, Journal of Asian Natural Products Research, 2021, 23(7): 692-702.
38. Tian Yuee, Sun Di, Han Xiaoxiao, Yang Jinming, Zhang Song, Feng Nannan, Zhu Lina, Xu Zhongyuan, Che Zhiping(通讯作者), Liu Shengming, Lin Xiaomin, Jiang Jia, Chen Genqiang, Synthesis, anti-oomycete activity, and SAR studies of paeonol derivatives, Journal of Asian Natural Products Research, 2021, 23(2): 138-149.
39. Che Zhiping(第一且通讯作者), Yang Jinming, Zhang Song, Sun Di, Tian Yuee, Liu Shengming, Lin Xiaomin, Jiang Jia, Chen Genqiang, Synthesis of novel 9R/S-acyloxy derivatives of cinchonidine and cinchonine as insecticidal agents, Journal of Asian Natural Products Research, 2021, 23(2): 163-175.
40. Che Zhiping(第一且通讯作者), Yang Jinming, Sun Di, Tian Yuee, Liu Shengming, Lin Xiaomin, Jiang Jia, Chen Genqiang, Synthesis of novel (9S)-acyloxy derivatives of quinidine and dihydroquinidine as insecticidal agents, Chemistry & Biodiversity, 2020, 17(4): e1900696.
41. Che Zhiping(第一且通讯作者), Yang Jinming, Sun Di, Tian Yuee, Liu Shengming, Lin Xiaomin, Jiang Jia, Chen Genqiang, Combinatorial synthesis of a series of paeonol-based phenylsulfonyl hydrazone derivatives as insecticidal agents, Combinatorial Chemistry & High Throughput Screening, 2020, 23(3): 232-238.
42. Che Zhiping(第一且通讯作者), Yang Jinming, Sun Di, Tian Yuee, Liu Shengming, Lin Xiaomin, Jiang Jia, Chen Genqiang, Combinatorial synthesis of novel 9R-acyloxyquinine derivatives as insecticidal agents, Combinatorial Chemistry & High Throughput Screening, 2020, 23(2): 111-118.
43. Chen Genqiang, Xia Yanfei, Yang Jinming, Che Zhiping(通讯作者), Sun Di, Li Shen, Tian Yuee, Liu Shengming, Jiang Jia, Lin Xiaomin, Controlled synthesis of N, N-dimethylarylsulfonamide derivatives as nematicidal agents, Journal of Asian Natural Products Research, 2020, 22(12): 1197-1206.
44. Tian Yuee, Sun Di, Yang Jinming, Che Zhiping(通讯作者), Liu Shengming, Lin Xiaomin, Jiang Jia, Chen Genqiang, Synthesis of sulfonate derivatives of maltol and their biological activity against Phytophthora capsici and Bursaphelenchus xylophilus in vitro, Journal of Asian Natural Products Research, 2020, 22(6): 578-587.
45. Che Zhiping(第一且通讯作者), Yang Jinming, Shan Xijie, Tian Yuee, Liu Shengming, Lin Xiaomin, Jiang Jia, Hu Mei, Chen Genqiang, Synthesis and insecticidal activity of sulfonate derivatives of sesamol against Mythimna separata in vivo, Journal of Asian Natural Products Research, 2020, 22(7): 678-688.
46. Che Zhiping(第一且通讯作者), Tian Yuee, Liu Shengming, Jiang Jia, Hu Mei, Chen Genqiang, Stereoselective synthesis of 4β-acyloxypodophyllotoxin derivatives as insecticidal agents, Journal of Asian Natural Products Research, 2019, 21(10): 1028-1041.
47. Che Zhiping(第一且通讯作者), Tian Yuee, Yang Jinming, Liu Shengming, Jiang Jia, Hu Mei, Chen Genqiang, Screening of insecticidal activity of podophyllotoxin analogues against Athetis dissimilis, Natural Product Communications, 2019, 14(1): 117-120.
48. Tian Yuee, Che Zhiping(共同第一作者), Sun Di, Yang Yuanyuan, Lin Xiaomin, Liu Shengming, Liu Xiaoyu, Gao Jie, Resistance identification of tree peony cultivars of different flowering time to gray mold pathogen Botrytis cinerea, HortScience, 2019, 54(2): 328-330.
49. Che Zhiping(第一作者), Tian Yuee, Liu Shengming, Hu Mei, Chen Genqiang, Discovery of N-arylsulfonyl-3-acylindole benzoyl hydrazine derivatives as anti-HIV-1 agents, Brazilian Journal of Pharmaceutical Sciences, 2018, 54(4): e17543.
50. Che Zhiping(第一作者), Tian Yuee, Liu Shengming, Hu Mei, Chen Genqiang, Synthesis and in vitro anti-HIV-1 evaluation of some N-arylsulfonyl-3-formylindoles, Brazilian Journal of Pharmaceutical Sciences, 2018, 54(3): e17044.
51. Che Zhiping(第一作者), Tian Yuee, Hu Zhenjie, Chen Yingwu, Liu Shengming, Chen Genqiang, Synthesis and in vitro anti-HIV-1 activity of a series of N-arylsulfonyl-3-propionylindoles, Zeitschrift für Naturforschung Section C-A Journal of Biosciences, 2016, 71(5-6)c: 105-109.
52. Che Zhiping(第一作者), Liu Shengming, Tian Yuee, Hu Zhenjie, Chen Yingwu, Chen Genqiang, Design and synthesis of novel N-arylsulfonyl-3-(2-yl-ethanone)-6-methylindole derivatives as inhibitors of HIV-1 replication, Pharmaceuticals (Basel), 2015, 8(2): 221-229.
53. Che Zhiping(第一作者), Yu Xiang, Fan Lingling, Xu, Hui, Insight into dihalogenation of E-ring of podophyllotoxins, and their acyloxyation derivatives at the C4 position as insecticidal agents, Bioorganic & Medicinal Chemistry Letters, 2013, 23(20): 5592-5598.
54. Che Zhiping(第一作者), Huang Ning, Yu Xiang, Yang Liumeng, Ran Junqiang, Zhi Xiaoyan, Xu Hui, Zheng Yongtang, Microwave-assisted combinatorial synthesis of 2-alkyl-2-(N-arylsulfonylindol-3-yl)-3-N-acyl-5-aryl-1,3,4-oxadiazolines as anti-HIV-1 agents, Combinatorial Chemistry & High Throughput Screening, 2013, 16(5): 400-407.
55. Che Zhiping(第一作者), Xu Hui, One-pot synthesis of dibenzofurans via SNAr and subsequent ligand-free palladium-catalyzed intramolecular aryl-aryl cross-coupling reactions under microwave irradiation, Zeitschrift für Naturforschung Section B-A Journal of Chemical Sciences, 2011, 66(8): 833-836.
56. 陈根强, 刘圣明, 车志平(通讯作者), 田月娥, 林晓民, 中国农药自主创制, 化学通报, 2020, 83(12): 1058-1080.
57. 杨进明, 陈根强, 田月娥, 刘圣明, 车志平(通讯作者), 丹皮酚类化合物及其生物活性研究进展, 化学通报, 2021, 84(8): 776-786.
58. 车志平(第一且通讯作者), 杨进明, 田月娥, 刘圣明, 姜佳, 陈根强, 奎宁类化合物研究进展, 化学通报, 2018, 81(9): 792-796+804.
59. 陈根强, 杨进明, 孙迪, 韩笑笑, 田月娥, 刘圣明, 姜佳, 车志平(通讯作者), 丹皮酚苯磺酰腙类衍生物的合成及杀粘虫活性研究, 化学通报, 2020, 83(2): 139-143.
60. 王瑞光, 魏如雪, 李岩, 田月娥, 车志平(通讯作者), 丹皮酚腙类化合物的合成及其杀虫活性研究, 现代农药, 2023, 22(6): 37-41+63.
61. 魏如雪, 李岩, 王瑞光, 田月娥, 黄晓博, 刘圣明, 陈根强, 车志平(通讯作者), 3种杀虫剂对牡丹刺蛾的田间防治效果, 世界农药, 2023, 45(7): 54-57.
62. 田月娥, 车志平(通讯作者), 刘圣明, 胡梅, 陈根强, N-苯磺酰基-3-酰基吲哚苯甲酰腙类化合物的抑菌活性, 农药, 2018, 57(4): 263-265.
63. 田月娥, 车志平(通讯作者), 刘圣明, 王华, 何虎, 胡梅, 陈根强, 几种醌类化合物抑菌活性研究, 农药, 2017, 56(11): 844-846.
64. 车志平(第一作者), 刘圣明, 魏素玲, 陈根强, 3-醛基吲哚类化合物的合成及对玉米大、小斑病菌的抑制作用, 农药, 2015, 54(03): 177-179.
65. 车志平(第一作者), 田月娥, 刘圣明, 崔林开, 徐建强, 魏素玲, 几种含羟基类化合物的抑菌活性,农药, 2015, 54 (12): 930-932+936.
六、发明专利
1. 车志平(1/7)等,9R-酰氧基奎宁类衍生物及其制备方法、奎宁或其衍生物的应用、植物源杀虫剂,2023-03-14,中国,授权专利号:ZL201911001679.5
2. 车志平(1/8)等, N, N-二甲基磺酰胺类衍生物的制备方法,2022-03-18,中国,授权专利号:ZL201910622055.9
3. 车志平(1/6)等,一种甲氧基苯乙酮衍生物及其制备方法、应用,2021-09-24,中国,授权专利号:ZL201710994239.9
4. 车志平(1/10)等,N, N-二甲基芳香基磺酰胺类衍生物及其在防治南方根结线虫方面的应用,2021-09-24,中国,授权专利号:ZL201910622062.9
5. 车志平(1/7)等,丹皮酚苯磺酰腙及其衍生物和其制备方法、植物源杀虫剂及其应用,2021-09-24,中国,授权专利号:ZL201910974310.6
6. 车志平(1/7)等,奎尼定或奎尼定类衍生物的应用、植物源杀虫剂、奎尼定类衍生物及其制备方法,2021-10-26,中国,授权专利号:ZL201911001717.7
7. 车志平(1/8)等,一种辛可尼丁类化合物及其制备方法、应用,杀虫剂,2020-10-02,中国,授权专利号:ZL201911002506.5
8. 车志平(1/8)等,二氢奎尼丁类化合物及其制备方法和应用、植物源杀虫剂,2020-10-02,中国,授权专利号:ZL201911002507.X
9. 车志平(1/5)等,磺酰基芝麻酚衍生物及其制备方法、农用杀虫剂、防治农业害虫方面的应用,2020-07-10,中国,授权专利号:ZL201910111754.7
10. 车志平(1/5)等, N-苯磺酰基-3-乙酰基吲哚酰腙类化合物、制备方法及应用,2019-02-26,中国,授权专利号:ZL201510597814.2
11. 车志平(1/5)等, N-苯磺酰基-3-(2-基-乙酰基)-6-甲基吲哚类衍生物的用途,2017-07-07,中国,授权专利号:ZL201510485923.5
12. 黄晓博,车志平(2/5)等,一种1-酰氧基芝麻酚类衍生物及其制备方法和应用,2024-02-27,中国,授权专利号:ZL202210755877.6
13. 董钧锋,车志平(2/7)等,一种丹皮酚腙类衍生物及其制备方法和应用、杀虫剂,2023-07-25,中国,授权专利号:ZL202011231908.5
14. 董钧锋,车志平(2/7)等,一种丹皮酚酰腙类衍生物及其制备方法和应用、杀虫剂,2023-05-09,中国,授权专利号:ZL202011233398.5
15. 陈根强,车志平(2/10)等,一种1-磺酰基萘酚类衍生物及其制备方法,2022-12-23,中国,授权专利号:ZL202011253857.6
16. 陈根强,车志平(2/8)等,一种9S-酰氧基辛可宁类衍生物及其制备方法和应用,植物源杀虫剂,2021-05-011,中国,授权专利号:ZL201911001699.2
17. 陈根强,车志平(2/10)等,一种1-磺酰基萘酚类衍生物在防治植物病原真菌中的应用、抗菌剂,2021-09-07,中国, 授权专利号:ZL202011253845.3
18. 田月娥,车志平(2/5)等,一种3-磺酰基麦芽酚衍生物及制备方法和应用,植物源杀菌剂,2021-03-16,中国,授权专利号:ZL201910110125.2
19. 陈根强,车志平(2/5)等,N-取代苯磺酰基-3-丙酰基吲哚类衍生物、制备方法及应用,2018-03-21,中国,授权专利号:ZL201510485695.1
20. 田月娥,车志平(2/5)等,噁唑啉类衍生物、制备方法及其在制备植物病原真菌抗菌剂方面的应用,2018-05-25,中国,授权专利号:ZL201510601292.9
21. 吕琪卉,田月娥,林丁,车志平(4/5)等,一种磺酰基桧木醇类衍生物及其制备方法和应用,2023-05-30,中国,授权专利号:ZL202210095254.0
七、成果奖励
1. 车志平(3/15),植物源农药新品创制与应用,河南省教育厅,科技成果奖,一等奖,2024;
2. 车志平(1/6),Stereoselective synthesis of 4β-acyloxypodophyllotoxin derivatives as insecticidal agents,河南省教育厅,优秀科技论文奖,二等奖,2021;
3. 车志平(10/10),设施果菜低碳绿色生产的根区调控关键技术开发与应用,河南省人民政府,河南省科学技术进步奖,二等奖,2020;
4. 车志平(6/9),天然产物结构优化及农用活性研究,陕西省人民政府,陕西省科学技术奖,二等奖,2018;
5. 车志平(5/7),设施蔬菜灰霉病抗药性分子检测及精准防控关键技术研究与应用,河南省人民政府,河南省科学技术进步奖,三等奖,2017;
6. 车志平(6/11),三种天然产物的结构优化及农用活性研究,陕西省教育厅,陕西高等学校科学技术奖,一等奖,2017;
7. 车志平(5/10),设施蔬菜灰霉病抗药性分子检测及精准防控关键技术研究与应用,河南省教育厅,科技成果奖,一等奖,2017。
八、教改成果
教改论文
1. 车志平(第一作者), 李秀珍, 田月娥, 以问题驱动与研讨为主的植物保护类研究生教学新模式研究, 高教学刊, 2023, 9: 113-116.
2. 车志平(第一作者),田月娥, 黄晓博, “植物化学保护学”课程教学新模式研究, 教育教学论坛, 2023, 42: 53-56.
3. 田月娥, 车志平(通讯作者), 基于学术创新能力提升的课程教学改革探索——以研究生课程“植物保护研究技术”为例, 教育教学论坛, 2023, 34: 104-108.
4. 车志平(第一作者), 陈应武, 普通高校科研与本科教学提升, 学园, 2015, 11: 25.
5. 陈应武, 胡镇杰, 车志平, 移动互联网技术在普通昆虫学教学中的应用实践, 学园, 2015, 11: 20-21.
教改项目
1. 以“面授、互联网与Seminar”相结合的研究生教学新模式研究: 以农药学硕士为例,河南科技大学,2020.01-2021.12,1.3万元,结题,主持;
2. 以“面授、互联网与Seminar”相结合的教学新模式研究:以植物化学保护课程为例,河南科技大学,2020.01-2021.12,1.0万元,结题,主持。
成果鉴定
1. 车志平(1/4),“面授、互联网与Seminar”相结合的教学新模式研究:以植物化学保护课程为例(HKDJGJT2023087),河南科技大学,2023;
2. 车志平(3/5),“农药生物测定”精品资源共享课程建设(2016YKJ-007),河南科技大学,2019。
九、竞赛获奖
1. 第十六届“挑战杯”河南省大学生课外学术科技作品竞赛,基于植物次生物质乙基麦芽酚和桧木醇的绿色杀菌剂创制研究,二等奖,指导教师,2023;
2. 第十四届“挑战杯”河南省大学生课外学术科技作品竞赛,小宗作物种苗期保护剂研究——绿豆和红豆保护剂(系列一),二等奖,指导教师,2019;
3. 第十届“挑战杯”河南科技大学大学生课外学术科技作品竞赛,基于植物次生物质乙基麦芽酚和桧木醇的绿色杀菌剂创制研究,一等奖,指导教师,2023;
4. 第八届“挑战杯”河南科技大学大学生课外学术科技作品竞赛,小宗作物种苗期保护剂研究——绿豆和红豆保护剂(系列一),一等奖,指导教师,2019。
十、培养学生
1. 邢濮厚,乙基麦芽酚磺酸酯类衍生物的合成及其抑菌活性研究,河南省优秀学士学位论文(毕业设计),指导教师,2024;
2. 邢濮厚,乙基麦芽酚和桧木醇磺酰氧基衍生物的合成及抑菌活性研究,国家级大学生创新训练计划重点支持领域项目(全校唯一),指导教师,2021;
3. 朱丽娜,熊果酸类衍生物的合成及其抑菌活性研究,硕士研究生国家奖学金,指导教师,2021;
4. 杨进明,丹皮酚酯与腙类衍生物的合成及农用生物活性研究,硕士研究生国家奖学金,指导教师,2020。
十一、服务社会
“服务基层需求,助推乡村振兴”,作为一名高校教师,职责所在,义不容辞。结合自身专业特色,助力河南省乡村振兴;充分发挥专业特长和科研优势,将专业特长和科研成果有机融合,更好服务河南省乡村振兴;以河南省和洛阳市科技特派员等项目为依托,重点围绕我省农作物主要病虫草害绿色防控关键技术,积极开展科技服务和培训。近三年,以办培训班、开现场会等多种形式普及科学技术,下乡科普近200人次;举办科普培训50多场,培训了30多个科技示范户和致富能手,培养了100多名农民技术人员,受训5000余人;发放图书1000余册,科普宣传资料5千余份,为我省农作物主要病虫草害绿色防控提供了有力的技术保障,切实做到了助农绿色增收。